EFTA00625099Set 9
30p10,397w
fold for PDE6, >80-fold for PDE1, >700-fold
for PDE2, PDE3, PDE4, PDE7, PDE8, PDE9, PDE1 0, and PDE11). The approximately
4,000-fold selectivity for PDE5 versus PDE3
https://www.justice.gov/epstein/files/DataSet%209/EFTA00625099.pdf